2-(4-氟苯基)噻唑-5-甲醛合成路线 (共 1 条)
反应条件
tetrakis(triphenylphosphine) palladium(0); sodium carbonate in ethanol; toluene T=85°C; 6 h; Inert atmosphere;
参考文献
ENDO PHARMACEUTICALS INC.; SMITH, Roger, Astbury; KETHIRI, Raghava, Reddy; KRISTAM, Rajendra; LAPING, Nicholas, James; VENKATESHAPPA, Chandregowda; KULKARNI, Bheemashankar; DEVRAJ, Rajesh; DEWANG, Purushottam
Patent: WO2013/49559 A1, 2013 ;
Location in patent: Page/Page column 52 ;