5-硝基-N-(4-(2-(吡咯烷-1-基)乙氧基)苯基)嘧啶-2-胺合成路线 （共 2 条）
反应条件
caesium carbonate; tris-(dibenzylideneacetone)dipalladium(0); 9,9-dimethyl-4,5-bis(diphenyl-phosphino)xanthene in 1,4-dioxane
2 - 18 h; Heating / reflux; Product distribution / selectivity;
参考文献
TARGEGEN, INC.
Patent: WO2008/8234 A1, 2008 ;
Location in patent: Page/Page column 61-62 ;
反应条件
hydrogen; palladium 10 on activated carbon in methanol
T=20°C; 1 - 2 h; Product distribution / selectivity;
参考文献
TARGEGEN, INC.
Patent: WO2008/8234 A1, 2008 ;
Location in patent: Page/Page column 62 ;
