反应条件
1: 74 percent / ethanol / Heating
2: 1) n-BuLi / 1) THF, hexane, -78 deg C, 5 min, 2) to -20 deg C
View Scheme
参考文献
Davis, Steven E.; Rauckman, Barbara S.; Chan, Joseph H.; Roth, Barbara
Journal of Medicinal Chemistry, 1989 , vol. 32, # 8 p. 1936 - 1942