hydrogenchloride; sodium hydroxide in ethanol 2 h; Heating;
参考文献
Das, Umashankar; Singh, Ravi S.P.; Alcorn, Jane; Hickman, Mark R.; Sciotti, Richard J.; Leed, Susan E.; Lee, Patricia J.; Roncal, Norma; Dimmock, Jonathan R.
Bioorganic and Medicinal Chemistry, 2013 , vol. 21, # 23 p. 7250 - 7256
potassium carbonate in N,N-dimethyl-formamide
T=100°C; 1.5 h;
参考文献
Jones, Charles D.; Jevnikar, Mary G.; Pike, Andrew J.; Peters, Mary K.; Black, Larry J.; at al.
Journal of Medicinal Chemistry, 1984 , vol. 27, # 8 p. 1057 - 1066