N-Boc-4-哌啶乙醇合成路线

参考文献

Nencini, Arianna; Castaldo, Cristiana; Comery, Thomas A.; Dunlop, John; Genesio, Eva; Ghiron, Chiara; Haydar, Simon; Maccari, Laura; Micco, Iolanda; Turlizzi, Elisa; Zanaletti, Riccardo; Zhang, Jean
European Journal of Medicinal Chemistry, 2014 , vol. 78, p. 401 - 418

89151-44-0N-Boc-4-哌啶乙醇

169457-73-24-(2-溴乙基)哌啶-1-羧酸叔丁酯

参考文献

AstraZeneca AB; NPS PHARMACEUTICALS
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US 20070032469 A1

558-13-4四溴化碳+

89151-44-0N-Boc-4-哌啶乙醇

169457-73-24-(2-溴乙基)哌啶-1-羧酸叔丁酯

参考文献

Glaxo Group Limited
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865-33-8甲醇钾+

89151-44-0N-Boc-4-哌啶乙醇

175213-46-41-N-BOC-4-哌啶乙酸甲酯

参考文献

Powell, Adam B.; Stahl, Shannon S.
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89151-44-0N-Boc-4-哌啶乙醇

114998-55-9

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Ambler, John; Brown, Lyndon; Cockcroft, Xiao-Ling; Gruetter, Markus; Hayler, Judy; Janus, Diana; Jones, Darryl; Kane, Peter; Menear, Keith; Priestle, John; Smith, Garrick; Talbot, Mark; Walker V, Clive; Wathey, Bernard
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89151-44-0N-Boc-4-哌啶乙醇+

74-88-4甲基碘

868849-54-14-甲氧基乙基哌啶盐酸盐

参考文献

Warner-Lambert Company LLC
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89151-44-0N-Boc-4-哌啶乙醇

885516-98-3

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Mi, Yuan; Corey
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89151-44-0N-Boc-4-哌啶乙醇

89151-46-24-(2-碘乙基)-1-哌啶羧酸叔丁酯

参考文献

Villalobos; Blake; Biggers; Butler; Chapin; Chen; Ives; Jones; Liston; Nagel; Nason; Nielsen; Shalaby; White
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288-32-4咪唑+

89151-44-0N-Boc-4-哌啶乙醇

89151-46-24-(2-碘乙基)-1-哌啶羧酸叔丁酯

参考文献

Merck and Co., Inc.
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89151-44-0N-Boc-4-哌啶乙醇+

98-59-9对甲苯磺酰氯

89151-46-24-(2-碘乙基)-1-哌啶羧酸叔丁酯

参考文献

Pfizer Inc.
Patent: US4489075 A1, 1984 ;