5-氯-6-吡嗪基-1-烟酸合成路线 (共 1 条)
反应条件
N-ethyl-N,N-diisopropylamine in N,N-dimethyl acetamide
T=120°C; 2 h;
参考文献
Bach, Peter; Bostroem, Jonas; Brickmann, Kay; Van Giezen; Groneberg, Robert D.; Harvey, Darren M.; O'Sullivan, Michael; Zetterberg, Fredrik
European Journal of Medicinal Chemistry, 2013 , vol. 65, p. 360 - 375