反应条件
1: 92 percent / 0.1N HCl / 0.17 h / 60 °C
2: 74 percent / Br2, sodium acetate / acetic acid / 1 h / Ambient temperature
3: 82 percent / KI, HCl / ethanol / 8 h / 100 °C
View Scheme
参考文献
Tarzia, Giorgio; Occelli, Emilio; Toja, Emilio; Barone, Domenico; Corsico, Nerina; et al.
Journal of Medicinal Chemistry, 1988 , vol. 31, # 6 p. 1115 - 1123