4-氯-3-(1-吡咯烷基羰基)苯硼酸合成路线 （共 2 条）
反应条件
1: With benzotriazol-1-ol; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride; N-ethyl-N,N-diisopropylamine in acetonitrile 2: With (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride; potassium acetate; 4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl-4',4',5',5'-tetramethyl-1,3,2-dioxaborolane in 2-methyl tetrahydrofuran 3: With hydrogenchloride; sodium periodate in 2-methyl tetrahydrofuran; water
参考文献
Zhu, Jason; Razler, Thomas M.; Xu, Zhongmin; Conlon, David A.; Sortore, Eric W.; Fritz, Alan W.; Demerzhan, Roman; Sweeney, Jason T.
Organic Process Research and Development, 2011 , vol. 15, # 2 p. 438 - 442
反应条件
1: With benzotriazol-1-ol; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride; N-ethyl-N,N-diisopropylamine in acetonitrile
2: With (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride; potassium acetate; 4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl-4',4',5',5'-tetramethyl-1,3,2-dioxaborolane in 2-methyl tetrahydrofuran
3: With hydrogenchloride; sodium periodate in 2-methyl tetrahydrofuran; water
参考文献
Zhu, Jason; Razler, Thomas M.; Xu, Zhongmin; Conlon, David A.; Sortore, Eric W.; Fritz, Alan W.; Demerzhan, Roman; Sweeney, Jason T.
Organic Process Research and Development, 2011 , vol. 15, # 2 p. 438 - 442
