反应条件
sodium cyanoborohydride; dimethyl sulfate 1.) ether, RT, 1 h, 2.) HMPA, 120 deg C, 16 h; Yield given. Multistep reaction;
参考文献
Hartmann, Rolf W.; Schwarz, Walter; Schoenenberger, Helmut
Journal of Medicinal Chemistry, 1983 , vol. 26, # 8 p. 1137 - 1144