N1,N4-双-Boc-亚精胺合成路线 （共 12 条）
反应条件
1: Et3N / CH2Cl2 / 0.17 h / -20 °C
2: aq. NH3 / ethanol / 48 h / Ambient temperature
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参考文献
Lebreton, Luc; Annat, Jocelyne; Derrepas, Philippe; Dutartre, Patrick; Renaut, Patrice
Journal of Medicinal Chemistry, 1999 , vol. 42, # 2 p. 277 - 290
反应条件
1: 100 percent / triethylamine / tetrahydrofuran / 24 h
2: 88 percent / K2CO , water / H2O; methanol / 2.17 h / Heating
View Scheme
参考文献
Bergeron, Raymond J.; McManis, James S.
Journal of Organic Chemistry, 1987 , vol. 52, # 9 p. 1700 - 1703
