反应条件
1: 2,3,5-tribromopyridine With n-butyllithium in diethyl ether
T=-78°C; 1.5 h;
2: N,N-dimethyl-formamide in diethyl ether
T=-78 - 20°C;
参考文献
Burzicki, Gregory; Voisin-Chiret, Anne Sophie; Santos, Jana Sopkova-De Oliveira; Rault, Sylvain
Synthesis, 2010 , # 16 art. no. T06810SS, p. 2804 - 2810