反应条件
tris-(dibenzylideneacetone)dipalladium(0); potassium carbonate; 9,9-dimethyl-4,5-bis(diphenyl-phosphino)xanthene in 1,4-dioxane
T=100°C; 16 h; Inert atmosphere;
参考文献
Kim, Se-Ho; Bajji, Ashok; Tangallapally, Rajendra; Markovitz, Benjamin; Trovato, Richard; Shenderovich, Mark; Baichwal, Vijay; Bartel, Paul; Cimbora, Daniel; McKinnon, Rena; Robinson, Rosann; Papac, Damon; Wettstein, Daniel; Carlson, Robert; Yager, Kraig M.
Journal of Medicinal Chemistry, 2012 , vol. 55, # 17 p. 7480 - 7501