6-溴-2-氟吡啶-3-胺合成路线 (共 1 条)
反应条件
1: With bromine; sodium acetate; acetic acid
T=0 - 5°C; 1 h;
2: With sodium hydroxide in water
T=0°C; pH=~ 5;
参考文献
AstraZeneca AB
Patent: US2008/221149 A1, 2008 ;
Location in patent: Page/Page column 22 ;
US 20080221149 A1