反应条件
1: 6N HCl / 5 h / Heating
2: 1.) n-BuLi / 1.) THF, hexane, -5 deg C, 2.) THF, hexane, 0 deg C, 2 h
View Scheme
参考文献
Bolhofer; Deana; Habecker; Hoffman; Gould; Pietruszkiewicz; Prugh; Torchiana; Cragoe Jr.; Hirschmann
Journal of Medicinal Chemistry, 1983 , vol. 26, # 4 p. 538 - 544