反应条件
1.1: 1,1-carbonyldiimidazole / tetrahydrofuran / 1.5 h / 20 °C 1.2: 2.50 g / NH3 / methanol; tetrahydrofuran / 0 - 20 °C 2.1: 38 percent / Lawesson's reagent / tetrahydrofuran / 3 h / Heating View Scheme
参考文献
Palmer, James T.; Bryant, Clifford; Wang, Dan-Xiong; Davis, Dana E.; Setti, Eduardo L.; Rydzewski, Robert M.; Venkatraman, Shankar; Tian, Zong-Qiang; Burrill, Leland C.; Mendonca, Rohan V.; Springman, Eric; McCarter, John; Chung, Tobee; Cheung, Harry; Janc, James W.; McGrath, Mary; Somoza, John R.; Enriquez, Philip; Yu, Z. Walter; Strickley, Robert M.; Liu, Liang; Venuti, Michael C.; Percival, M. David; Falgueyret, Jean-Pierre; Prasit, Peppi; Oballa, Renata; Riendeau, Denis; Young, Robert N.; Wesolowski, Gregg; Rodan, Sevgi B.; Johnson, Colena; Kimmel, Donald B.; Rodan, Gideon
Journal of Medicinal Chemistry, 2005 , vol. 48, # 24 p. 7520 - 7534