反应条件
1: 1.) NaH / 1.) DMF, 30 min, 2.) DMF, 60 deg C, 10 h 2: NaN3, NaI, 18-crown-6 / dimethylformamide / 18 h / 60 °C View Scheme
参考文献
Bhagwat; Gude; Boswell; Contardo; Cohen; Dotson; Mathis; Lee; Furness; Zoganas
Journal of Medicinal Chemistry, 1992 , vol. 35, # 23 p. 4373 - 4383