反应条件
1: 4-(6-fluoro-1,2-benzisoxazol-3-yl)-piperidine With potassium carbonate; potassium iodide in acetonitrile T=30 - 60°C; 2: (±)-3-(2-chloroethyl)-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one monohydrochloride in acetonitrile 47 h;
参考文献
CADILA PHARMACEUTICALS LTD.; SODAGAR, Keval, Rameshchandra; MALIK, Vineet; DESAI, Bharat, Ramchandra; JAIN, Sudhir, Hukamchand; PARIKH, Sanjay, Natvarlal; SHARMA, Arun, Omprakash; BAPAT, Uday, Rajaram; KHAMAR, Bakulesh, Mafatlal
Patent: WO2010/82111 A1, 2010 ;
Location in patent: Page/Page column 8-9 ;