2-氨基-3-氟苯甲酸合成路线

825-22-92-氨基-3-氟苯甲酸

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108665-36-7

参考文献

Cosmo, Robert; Sternhell, Sever
Australian Journal of Chemistry, 1987 , vol. 40, # 1 p. 35 - 47

825-22-92-氨基-3-氟苯甲酸

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387-48-43-氟-2-碘苯甲酸

参考文献

Uchikawa, Osamu; Mitsui, Keita; Asakawa, Akiko; Morimoto, Shigeru; Yamamoto, Masataka; Kimura, Hiroyuki; Moriya, Takeo; Mizuno, Masahiro
Patent: US2003/187014 A1, 2003 ;

825-22-92-氨基-3-氟苯甲酸

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348-54-92-氟苯胺

参考文献

Hooker Chemicals and Plastics Corp.
Patent: US4343951 A1, 1982 ;

825-22-92-氨基-3-氟苯甲酸

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187805-54-52-氨基-3-氟苯甲酰胺

参考文献

Hadd, Michael J.; Holladay, Mark W.; Rowbottom, Martin
Patent: US2012/53174 A1, 2012 ;
Location in patent: Page/Page column 49 ;
US 20120053174 A1

825-22-92-氨基-3-氟苯甲酸+

57-13-6尿素

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959236-96-58-氟-2,4(1H,3H)-喹唑啉二酮

参考文献

RANBAXY LABORATORIES LIMITED; DAS, Biswajit; UPADHYAY, Dilip, J.; PURNAPATRE, Kedar; GHOSH, Soma; KATOCH, Rita
Patent: WO2012/14109 A1, 2012 ;
Location in patent: Page/Page column 14 ;
WO 2012/014109 A1

590-28-3氰酸钾+

825-22-92-氨基-3-氟苯甲酸

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959236-96-58-氟-2,4(1H,3H)-喹唑啉二酮

参考文献

Ife, Robert J.; Brown, Thomas H.; Blurton, Peter; Keeling, David J.; Leach, Colin A.; et al.
Journal of Medicinal Chemistry, 1995 , vol. 38, # 14 p. 2763 - 2773

590-28-3氰酸钾+

825-22-92-氨基-3-氟苯甲酸

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959237-64-02,4-二氯-8-氟喹唑啉

参考文献

Clasby, Martin C.; Chackalamannil, Samuel; Stamford, Andrew
Patent: US2008/255156 A1, 2008 ;
Location in patent: Page/Page column 10 ;

825-22-92-氨基-3-氟苯甲酸

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959237-64-02,4-二氯-8-氟喹唑啉

参考文献

Thorat, Dhanaji Achyutrao; Doddareddy, Munikumar Reddy; Seo, Seon Hee; Hong, Tae-Joon; Cho, Yong Seo; Hahn, Ji-Sook; Pae, Ae Nim
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 6 p. 1593 - 1597

825-22-92-氨基-3-氟苯甲酸+

74-89-5甲胺

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1017789-26-22-氨基-3-氟-N-甲基-苯甲酰胺

参考文献

ASTRAZENECA AB; ASTRAZENECA UK LIMITED
Patent: WO2009/153589 A1, 2009 ;
Location in patent: Page/Page column 149 ;
WO 2009/153589 A1

825-22-92-氨基-3-氟苯甲酸

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1000339-91-22-溴-3-氟苯甲酰氯

参考文献

McKittrick, Brian; Failli, Amedeo; Steffan, Robert J.; Soll, Richard M.; Hughes, Philip; et al.
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