反应条件
1: 4,9-dihydro-3H-pyrido[3,4-b]indole With sodium hydride in N,N-dimethyl-formamide
T=-10°C; 1 h;
2: methyl 4-toluenesulfonate in N,N-dimethyl-formamide
T=-60°C; 2 h;
参考文献
Bertrand, Martial; Poissonnet, Guillaume; Theret-Bettiol, Marie-Helene; Gaspard, Christiane; Werner, Georges H.; Pfeiffer, Bruno; Renard, Pierre; Leonce, Stephane; Dodd, Robert H.
Bioorganic and Medicinal Chemistry, 2001 , vol. 9, # 8 p. 2155 - 2164
