反应条件
1: 96 percent / K2CO3, Cu, coprous oxide / 2-ethoxy-ethanol / 0.5 h / 120 °C
2: 41 percent / conc. H2SO4 / 2 h / 90 °C
3: pyridine, PCl3 / Heating
4: SOCl2, DMF / 0.5 h / Heating
View Scheme
参考文献
Denny; Atwell; Baguley
Journal of Medicinal Chemistry, 1983 , vol. 26, # 11 p. 1619 - 1625