Antonios-McCrea, William R.; Frazier, Kelly A.; Jazan, Elisa M.; Machajewski, Timothy D.; McBride, Christopher M.; Pecchi, Sabina; Renhowe, Paul A.; Shafer, Cynthia M.; Taylor, Clarke
Tetrahedron Letters, 2006 , vol. 47, # 5 p. 657 - 660
1: With hydrogen bromide; sodium nitrite in 1,4-dioxane; water T=0°C; 3 h; 2: With hydrogen bromide; copper(I) bromide in 1,4-dioxane; water T=0 - 50°C; 0.583333 h;
参考文献
MERCK SHARP and DOHME LIMITED
Patent: WO2003/99816 A1, 2003 ;
Location in patent: Page 58 ;
WO 03/099816 A1