mercury(II) diacetate in tetrahydrofuran T=60°C; 3 h;

1: sodium hydroxide; water / methanol / 5 h / 0 - 20 °C 2: 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride; benzotriazol-1-ol / N,N-dimethyl-formamide / 24 h / 20 °C 3: toluene-4-sulfonic acid / methanol / 12 h / 20 °C 4: copper(II) sulfate; TBTA; sodium L-ascorbate / water; methanol / 24 h / 20 °C / |Combinatorial reaction / High throughput screening (HTS) View Scheme

water; sodium hydroxide in methanol T=0 - 20°C; 5 h;

methanol; potassium carbonate T=20°C; 0.0833333 h;