反应条件
1: With potassium hydroxide; tris-(dibenzylideneacetone)dipalladium(0); di-tert-butyl(2′,4′,6′-triisopropylbiphenyl-2-yl)phosphine in 1,4-dioxane; water
T=100°C; 2 h;
2: With hydrogenchloride in 1,4-dioxane; water
参考文献
SCHERING CORPORATION; SHIPPS, JR., Gerald, W.; CHENG, Cliff, C.; HUANG, Xiaohua; ACHAB, Abdelghani, Abe; ORTH, Peter; VOIGT, Johannes, H.; SOUCY, Kyle, Ann
Patent: WO2010/56631 A1, 2010 ;
Location in patent: Page/Page column 123 ;
WO 2010/056631 A1