1: 73 percent / DMAP, DCC / CH2Cl2 / 4 °C 2: 89 percent / H2 / Pd / methanol / 4 h 3: 82 percent / Et3N / H2O / 1 h / Ambient temperature View Scheme
参考文献
Okada, Yoshio; Iguchi, Shin
Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1988 , p. 2129 - 2136
Barton, Derek H. R.; Crich, David
Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1986 , p. 1603 - 1612