反应条件
1: 1.) DME, ice bath, 1 h, 2.) EtOH, reflux, 2 h, 3.) Na2CO3
2: 1N NaOH / ethanol; H2O / 0.5 h / Heating
View Scheme
参考文献
Ager; Barnes; Danswan; Hairsine; Kay; Kennewell; Matharu; Miller; Robson; Rowlands; Tully; Westwood
Journal of Medicinal Chemistry, 1988 , vol. 31, # 6 p. 1098 - 1115