反应条件
diphenylphosphoranyl azide; triethylamine in N,N-dimethyl-formamide
1.) -20 deg C, 1 h, 2.) 20 deg C, 20 h;
参考文献
Montgomery, John A.; Thomas, H. Jeanette; Brockman, R. Wallace; Wheeler, Glynn P.
Journal of Medicinal Chemistry, 1981 , vol. 24, # 2 p. 184 - 189