反应条件
1: 1.) n-BuLi / 1.) THF, hexane, 0 deg C, 20 min, 2.) THF, RT, 24 h
2: 75 percent / KOH / methanol; H2O / 0.5 h / Heating
View Scheme
参考文献
Dawson, Marcia I.; Chan, Rebecca L.-S.; Derdzinski, Krzysztof; Hobbs, Peter D.; Chao, Wan-Ru; Schiff, Leonard J.
Journal of Medicinal Chemistry, 1983 , vol. 26, # 11 p. 1653 - 1656