1: With sodium acetate; sodium tris(acetoxy)borohydride in dichloromethane T=20°C; 16 h; 2: With sodium hydroxide; water; sodium hydrogencarbonate in dichloromethane Product distribution / selectivity;
参考文献
CYCLACEL LIMITED
Patent: WO2009/40556 A1, 2009 ;
Location in patent: Page/Page column 44; 75 ;
WO 2009/040556 A1