反应条件
1: With Rink amide resin; benzotriazol-1-ol; O-(benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium tetrafluoroborate; N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide T=0 - 20°C; 3.5 h; 2: With piperidine in N,N-dimethyl-formamide T=20°C; 0.416667 h; 3: With trifluoroacetic acid
参考文献
Tetrahedron, , vol. 58, # 28 p. 5741 - 5746