反应条件
1: With diphenyl phosphoryl azide; triethylamine in N,N-dimethyl-formamide T=20°C; 3 h; 2: With water in N,N-dimethyl-formamide T=100°C; 1 h;
参考文献
ABBOTT LABORATORIES; ROCKWAY, Todd W.; BETEBENNER, David A.; DEGOEY, David A.; FLENTGE, Charles A.; HUTCHINSON, Douglas K.; KATI, Warren M.; KRUEGER, Allan C.; LIU, Dachun; LONGENECKER, Kenton L.; PRATT, John K.; STEWART, Kent D.; WAGNER, Rolf
Patent: WO2010/111437 A1, 2010 ;
Location in patent: Page/Page column 74 ;
WO 2010/111437 A1