反应条件
1: 77 percent / sodium borohydride / methanol; H2O / 2 h / Ambient temperature
2: 1.) sodium hydride / 1.) DMF, r.t.; 2.) DMF, 2 h, r.t.
View Scheme
参考文献
Cozzi; Pillan; Bertone; et al.
European Journal of Medicinal Chemistry, 1985 , vol. 20, # 3 p. 241 - 245