反应条件
1: isopropyl alcohol / 20 h / |Reflux 2: lithium hydroxide hydrate; water / 24 h / 20 °C 3: (benzotriazo-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate / N,N-dimethyl-formamide / 24 h / 20 °C View Scheme
参考文献
Marson, Charles M.; Matthews, Christopher J.; Yiannaki, Elena; Atkinson, Stephen J.; Soden, Peter E.; Shukla, Lena; Lamadema, Nermina; Thomas, N. Shaun B.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 15 p. 6156 - 6174