联硼酸频那醇酯合成路线

参考文献

ASTRAZENECA AB; ASTEX THERAPEUTICS LTD
Patent: WO2007/145571 A1, 2007 ;
Location in patent: Page/Page column 88 ;
WO 2007/145571 A1

1188322-48-6+

73183-34-3联硼酸频那醇酯

1188322-50-0+

97728-11-5

参考文献

Inglis, Steven R.; Zervosen, Astrid; Woon, Esther C. Y.; Gerards, Thomas; Teller, Nathalie; Fischer, Delphine S.; Luxen, Andre; Schofield, Christopher J.
Journal of Medicinal Chemistry, 2009 , vol. 52, # 19 p. 6097 - 6106

3279-90-16-溴-1,2,3,4-四氢-2-喹啉酮+

73183-34-3联硼酸频那醇酯

400620-72-66-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-3,4-二氢喹啉-2(1H)-酮

参考文献

F. HOFFMANN-LA ROCHE AG; HOFFMANN-LA ROCHE INC.; CHENG, Zhanling; HAN, Xingchun; JIANG, Min; WANG, Jianhua; WANG, Min; YANG, Song; ZHOU, Chengang
Patent: WO2014/90692 A1, 2014 ;
Location in patent: Page/Page column 64 ;

425378-78-5+

73183-34-3联硼酸频那醇酯

425378-79-6

参考文献

Carling, William Robert; Hallett, David James; Russell, Michael Geoffrey Neil; Street, Leslie Joseph
Patent: US2003/55060 A1, 2003 ;

425378-77-4+

73183-34-3联硼酸频那醇酯

425378-79-6

参考文献

Jennings, Andrew S.R.; Lewis, Richard T.; Russell, Michael G.N.; Hallett, David J.; Street, Leslie J.; Castro, Jose L.; Atack, John R.; Cook, Susan M.; Lincoln, Rachael; Stanley, Joanna; Smith, Alison J.; Reynolds, David S.; Sohal, Bindi; Pike, Andrew; Marshall, George R.; Wafford, Keith A.; Sheppard, Wayne F.A.; Tye, Spencer J.
Bioorganic and Medicinal Chemistry Letters, 2006 , vol. 16, # 6 p. 1477 - 1480

475272-13-0

参考文献

Hamilton, Andrew D.; Ernst, Justin; Orner, Brendan P.
Patent: US2003/8882 A1, 2003 ;

79669-50-42-甲基-5-溴苯甲酸甲酯+

73183-34-3联硼酸频那醇酯

478375-39-22-甲基-5-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)苯甲酸甲酯

参考文献

Imanishi, Masashi; Nakajima, Yutaka; Tomishima, Yasuyo; Hamashima, Hitoshi; Washizuka, Kenichi; Sakurai, Minora; Matsui, Shigeo; Imamura, Emiko; Ueshima, Koji; Yamamoto, Takao; Yamamoto, Nobuhiro; Ishikawa, Hirofumi; Nakano, Keiko; Unami, Naoko; Hamada, Kaori; Matsumura, Yasuhiro; Takamura, Fujiko; Hattori, Kouji
Journal of Medicinal Chemistry, 2008 , vol. 51, # 15 p. 4804 - 4822

150529-73-02-(3-溴苯基)乙酸甲酯+

73183-34-3联硼酸频那醇酯

478375-42-7

参考文献

Kranich, Remo; Busemann, Anke S.; Bock, Daniel; Schroeter-Maas, Sabine; Beyer, Diana; Heinemann, Bo; Meyer, Michael; Schierhorn, Katrin; Zahlten, Rainer; Wolff, Gerhard; Aydt, Ewald M.
Journal of Medicinal Chemistry, 2007 , vol. 50, # 6 p. 1101 - 1115

73183-34-3联硼酸频那醇酯+

147283-87-2

478375-42-7

参考文献

Robichaud, Joel; Oballa, Renata; Prasit, Peppi; Falgueyret, Jean-Pierre; Percival, M. David; Wesolowski, Gregg; Rodan, Sevgi B.; Kimmel, Donald; Johnson, Colena; Bryant, Cliff; Venkatraman, Shankar; Setti, Eduardo; Mendonca, Rohan; Palmer, James T.
Journal of Medicinal Chemistry, 2003 , vol. 46, # 17 p. 3709 - 3727

294860-58-5+

73183-34-3联硼酸频那醇酯

478375-44-9

参考文献

AMIRA PHARMACEUTICALS, INC.
Patent: WO2009/108720 A2, 2009 ;
Location in patent: Page/Page column 119 ;
WO 2009/108720 A2