反应条件
1: 6-amino-1-benzyl-1,3-dihydropyrimidine-2,4-dione With bromine; sodium hydrogencarbonate in methanol T=0 - 20°C; 0.5 h; 2: methylamine in methanol; water T=70°C; 4 h;
参考文献
Alphey, Magnus S.; Pirrie, Lisa; Torrie, Leah S.; Boulkeroua, Wassila Abdelli; Gardiner, Mary; Sarkar, Aurijit; Maringer, Marko; Oehlmann, Wulf; Brenk, Ruth; Scherman, Michael S.; McNeil, Michael; Rejzek, Martin; Field, Robert A.; Singh, Mahavir; Gray, David; Westwood, Nicholas J.; Naismith, James H.
ACS Chemical Biology, 2013 , vol. 8, # 2 p. 387 - 396