4,6-二氯-2-三氟甲基嘧啶合成路线 (共 2 条)
反应条件
trichlorophosphate in water; triethylamine
反应条件
N-ethyl-N,N-diisopropylamine in tetrahydrofuran T=20°C; 60 h;
参考文献
TAISHO PHARMACEUTICAL CO., LTD.; Arena Pharmaceuticals, Inc
Patent: WO2005/95357 A2, 2005 ;
Location in patent: Page/Page column 140; 141 ;
WO 2005/095357 A2