1: With lithium aluminium tetrahydride in tetrahydrofuran T=0 - 20°C; 1 h; 2: With ethyl acetate in tetrahydrofuran 3: With sodium hydroxide; water in tetrahydrofuran
参考文献
ASTRAZENECA AB; ASTRAZENECA UK LIMITED
Patent: WO2005/61465 A1, 2005 ;
Location in patent: Page/Page column 62 ;
WO 2005/061465 A1