反应条件
1: oxalyl dichloride / dichloromethane; N,N-dimethyl-formamide / 24 h / 20 °C 2: N-ethyl-N,N-diisopropylamine / N,N-dimethyl-formamide / 24 h / 20 °C 3: triethylamine / methanol / 33 °C View Scheme
参考文献
Ochiana, Stefan O.; Pandarinath, Vidya; Wang, Zhouxi; Kapoor, Rishika; Ondrechen, Mary Jo; Ruben, Larry; Pollastri, Michael P.
European Journal of Medicinal Chemistry, 2013 , vol. 62, p. 777 - 784