反应条件
1: acetonitrile / 0.25 h / 200 °C / |Microwave irradiation
2: sodium methylate / N,N-dimethyl-formamide / 0.25 h / 200 °C / |Microwave irradiation
3: hydrogen; palladium on activated charcoal / tetrahydrofuran; methanol / 0.83 h
View Scheme
参考文献
Harusawa, Shinya; Sawada, Koichi; Magata, Takuji; Yoneyama, Hiroki; Araki, Lisa; Usami, Yoshihide; Hatano, Kouta; Yamamoto, Kouichi; Yamamoto, Daisuke; Yamatodani, Atsushi
Bioorganic and Medicinal Chemistry Letters, 2013 , vol. 23, # 23 p. 6415 - 6420