反应条件
1: With hydrogenchloride in 1,4-dioxane Reflux; 2: With sodium hydrogencarbonate in 1,4-dioxane; methanol; water T=20°C;
参考文献
TEXAS HEART INSTITUTE; BIEDIGER, Ronald, J.; GUNDLACH, IV, C., William; MARKET, Robert, V.; SAVAGE, Michael, M.; VANDERSLICE, Peter
Patent: WO2012/68251 A2, 2012 ;
Location in patent: Page/Page column 56 ;