1: With toluene-4-sulfonic acid T=60°C; 2: With lithium aluminium tetrahydride in tetrahydrofuran T=0 - 20°C; 2 h; 3: With water; ethyl acetate in tetrahydrofuran
参考文献
GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES; SOUTH ALABAMA MEDICAL SCIENCE FOUNDATION
Patent: WO2009/6089 A2, 2009 ;
Location in patent: Page/Page column 21 ;
WO 2009/006089 A2