反应条件
1: C5H8O2(2-)*2Li(1+) With N,N'-dimethyl-N,N'-propyleneurea in tetrahydrofuran T=5°C; 0.5 h; 2: ethyl iodide in tetrahydrofuran T=20°C; 2 h;
参考文献
Kaufmann, Dan; Bialer, Meir; Shimshoni, Jakob Avi; Devor, Marshall; Yagen, Boris
Journal of Medicinal Chemistry, 2009 , vol. 52, # 22 p. 7236 - 7248