反应条件
1: 1.) thionyl chloride, 2.) aq. ammonia / 1.) toluene, reflux, 1 h, 2.) toluene, 3 h
2: 60 percent / acetic acid / 20 h / Ambient temperature
View Scheme
参考文献
Pentassuglia, Giorgio; Bertani, Barbara; Donati, Daniele; Ursini, Antonella
Journal of Heterocyclic Chemistry, 1996 , vol. 33, # 4 p. 1163 - 1170