2-[[1-[7-甲基-2-(吗啉-4-基)-4-氧代-4H-吡啶并[1,2-a]嘧啶-9-基]乙基]氨基]苯甲酸合成路线 （共 1 条）
反应条件
1: 9-(1-hydroxyethyl)-7-methyl-2-morpholin-4-yl-4H-pyrido[1,2-a]pyrimidin-4-one With phosphorus tribromide in dichloromethane
T=40°C; 2.5 h;
2: anthranilic acid With triethylamine in dichloromethane
T=40°C;
3: With hydrogenchloride; water in acetone
T=20°C;
参考文献
Fjellstrom, Ola; Gustafsson, David; Lindberg, Jan A.; Jackson, Shaun
Patent: US2009/191177 A1, 2009 ;
Location in patent: Page/Page column 7 ;
US 20090191177 A1
