1: 17.5 percent / diphenyl phosphorazidate, NEt3 / 5 h / Heating
2: trifluoroacetic acid / 0.25 h
View Scheme
参考文献
Hardy, George W.; Lowe, Lawrence A.; Mills, Gail; Sang, Pang Yih; Simpkin, Dean S. A.; et al.
Journal of Medicinal Chemistry, 1989 , vol. 32, # 5 p. 1108 - 1118
