反应条件
1: sodium azide, NaI / dimethylformamide / 18 h / 60 °C 2: 1.) Ph3P, 2.) H2O / 1.) THF, RT, 10 h, 2.) THF, RT, 24 h View Scheme
参考文献
Maduskuie, Thomas P.; Wilde, Richard G.; Billheimer, Jeffrey T.; Cromley, Debra A.; Germain, Sandra; et al.
Journal of Medicinal Chemistry, 1995 , vol. 38, # 7 p. 1067 - 1083