3-[苯基-(甲苯-4-磺酰基)-氨基]-丙酸合成路线 (共 14 条)
反应条件
1: phosphorus oxychloride 2: methanol / 140 °C View Scheme
参考文献
Backeberg
Journal of the Chemical Society, 1933 , p. 618
反应条件
1: 1.) PCl5, 2.) AlCl3 / 1.) benzene, from 5 deg C to 23 deg C, 30 min, 2.) benzene 15-20 deg C, 3.5 h 2: 83 percent / gl. AcOH, aq. HCl / 3.5 h / Heating View Scheme
参考文献
Hueckel; Hagedorn
Chemische Berichte, 1957 , vol. 90, p. 752
参考文献
Journal of the Chemical Society, , vol. 125, p. 1618
参考文献
Clemo; Perkin
Journal of the Chemical Society, 1924 , vol. 125, p. 1618
Full Text Show Details
Backeberg
Journal of the Chemical Society, 1933 , p. 618
参考文献
Clemo; Perkin
Journal of the Chemical Society, 1924 , vol. 125, p. 1618
Full Text Show Details
Backeberg
Journal of the Chemical Society, 1933 , p. 618
反应条件
1: phosphorus oxychloride 2: acetic acid View Scheme
参考文献
Backeberg
Journal of the Chemical Society, 1933 , p. 618
参考文献
Takata
Yakugaku Zasshi, 1952 , vol. 72, p. 321
Chem.Abstr., 1953 , p. 2129
参考文献
Johnson; Woroch; Buell
Journal of the American Chemical Society, 1949 , vol. 71, p. 1901,1905
反应条件
1: pyridine / 0.33 h / Heating
2: aq. HCl / dioxane / 3 h / Heating
View Scheme
参考文献
Werbel, L. M.; Kesten, S. J.; Turner, W. R.
European Journal of Medicinal Chemistry, 1993 , vol. 28, # 11 p. 837 - 852
反应条件
1: acetic acid
2: pyridine
3: aqueous methanol. KOH-solution
View Scheme
参考文献
Johnson; Woroch; Buell
Journal of the American Chemical Society, 1949 , vol. 71, p. 1901,1905