1: With hydrogenchloride; hydrogen; palladium(II) hydroxide/carbon in ethanol; water
P=2585.81 Torr; 8 h;
2: With sodium hydrogencarbonate in water
pH=8 - 9;
参考文献
TARGACEPT, INC.
Patent: WO2006/23630 A2, 2006 ;
Location in patent: Page/Page column 63 ;