N-(吡啶-2-基)苯并[d]噁唑-2-胺合成路线 （共 2 条）
反应条件
1: With caesium carbonate; 9,9-dimethyl-4,5-bis(diphenyl-phosphino)xanthene in 1,4-dioxane
0.166667 h; Inert atmosphere;
2: With tris-(dibenzylideneacetone)dipalladium(0) in 1,4-dioxane
T=90°C; 30 h;
参考文献
KARUS THERAPEUTICS LTD; SHUTTLEWORTH, Stephen Joseph; TOMASSI, Cyrille Davy; CECIL, Alexander Richard Liam; MACCORMICK, Somhairle; NODES, William John; SILVA, Franck Alexandre
Patent: WO2014/72714 A1, 2014 ;
Location in patent: Page/Page column 35 ;
反应条件
in water
T=100°C; 16 h;
参考文献
Sycheva,T.P. et al.
Chemistry of Heterocyclic Compounds (New York, NY, United States), 1966 , vol. 2, p. 144 - 148
Khimiya Geterotsiklicheskikh Soedinenii, 1966 , vol. 2, p. 205 - 211
