potassium tert-butylate in tetrahydrofuran; tert-butyl alcohol
T=0 - 20°C; Henry reaction; 24 h;
参考文献
Gorczynski, Michael J.; Smitherman, Pamela K.; Akiyama, Taro E.; Wood, Harold B.; Berger, Joel P.; King, S. Bruce; Morrow, Charles S.
Journal of Medicinal Chemistry, 2009 , vol. 52, # 15 p. 4631 - 4639