1: thionyl chloride / DMF / CH2Cl2 / 20 h / 20 °C
2: 280 mg / pyridine / CH2Cl2 / 3 h / 0 °C
View Scheme
参考文献
Zhang, Jianmin; Pettersson, Hanna I.; Huitema, Carly; Niu, Chunying; Yin, Jiang; James, Michael N. G.; Eltis, Lindsay D.; Vederas, John C.
Journal of Medicinal Chemistry, 2007 , vol. 50, # 8 p. 1850 - 1864